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杨碧娟

发布日期:2022-04-21    作者:     来源:     点击:

基本情况

姓名: 杨碧娟

学历: 博士研究生

职务:

通信地址:云南民族大学呈贡校区民族医药学院

职称: 讲师

学位: 博士

电子邮箱:1940726755@126.com

邮编:650504

教育经历

2018年-2021年,中国科学院大学昆明植物研究所药物化学专业博士研究生

2015年-2018年,云南大学有机化学专业硕士研究生

2011年-2015年,云南师范大学制药工程专业本科

研究方向及招生专业

研究方向:天然产物先导化合物发现,活性分子结构修饰

招生专业:药学、化学生物学

教学工作

药物设计与筛选、天然药物化学实验

学术论文与著作

[1] Yang Bi-juan; Fan Shi-rui; Cai Jie-yun; Wang Yi-ting; Iing Chen-xu; Guo Jing-jing; Chen Duo-zhi; Hao Xiao-jiang; Aphananoid A is an Anti-Inflammatory Limonoid with a New 5/6/5 Fused Ring Featuring a C24 Carbon Skeleton from Aphanamixis polystachya. J Org Chem. 2020. 85(13): 8597-8602.

[2] Yang Bi-juan; Fan Shi-rui; Zhang Xin-fang; Cai Jie-yun; Ruan Ting; Xiang Zheng-rui; Ren Juan; Hao Xiao-jiang; Chen Duo-zhi; Design, synthesis and structure-activity relationship optimization of phenanthridine derivatives as new anti-vitiligo compounds, Bioorg Chem. 2022, 119: 105582.

[3] Chen Duo-zhi﹟; Yang Bi-juan﹟; He Xiao-li; Fan Shi-rui; Cai Jie-yun; Jing Chen-xu; Zhang Heng; Zhang Yu; Li Lin; Hao Xiao-jiang; Design, synthesisand structure-activity relationship optimization of phenanthridine derivatives as new Wnt/β-catenin signalling pathway Agonists, Bioorg Chem. 2018. 84: 285-294.

[4] Chen Duo-zhi; Zhang Heng; Jing Chen-xu; He Xiao-li; Yang Bi-juan; Cai Jie-yun; Zhou Yun-fu; Song Xiao-ming; Li Lin; Hao Xiao-jiang; Efficient synthesis of new phenanthridine Wnt/β-catenin signaling pathway agonists, Eur J Med Chem. 2018, 157: 1499.

[5] Wang Yi-ting; Long Xin-yan; Ding xiao; Fan Shi-rui; Cai Jie-yun; Yang Bi-juan; Zhang Xin-fang; Luo Rong-hua; Yang Lian; Ruan Ting; Ren Juan; Jing Chen-xu; Zheng Yong-tang; Hao Xiao-jiang; Chen Duo-zhi; Novel nucleocapsid protein-targeting phenanthridine inhibitors of SARS-CoV-2, European Journal of Medicinal Chemistry. Eur J Med Chem. 2022, 227: 113966.

[6] Chen Duo-Zhi; Fan Shi-Rui; Yang Bi-Juan; Yao Huo-Chun; Wang Yi-Ting; Cai Jie-Yun; Jing Chen-xu; Pao Zi-Hao; Luo Miao; Yuze Yan-Qiu; Liu Guang-Jin; Hao Xiao-jiang; Phenanthridine Derivative Host Heat Shock Cognate 70 Down-Regulators as Porcine Epidemic Diarrhea Virus Inhibit. J. Nat. Prod. 2021, 84, 1175−1184.

[7] Wang Yi-Ting; Fan Shi-Rui; Cai Jie-Yun; Guo Jing-Jing; Zhang Xin-Fang; Yang Bi-Juan; Hao Xiao-Jiang; Chen Duo-Zhi; Two new cytotoxic cycloartane triterpenoids from Aphanamixis polystachya (Wall.) R. N, Parker, Nat Prod Res. 2021: 1-6.

[8] Fan Shi-Rui; Guo Jing-Jing; Wang Yi-Ting; Yang Bi-Juan; Chen Duo-Zhi; Hao Xiao-Jiang; Two new bioactive lignans from leaves and twigs of Cleistanthus concinnus Croizat, Nat Prod Res. 2020, 34(23): 3328-3334.

[9] Jing Chen-Xu; Guo Jing-Jing; Yang Bi-Juan; Fan Shi-Rui; Wang Yi-Ting; Chen Duo-Zhi; Hao Xiao-Jiang; Stelleraguaianone B and C, two new sesquiterpenoids from Stellera chamaejasme L, Fitoterapia. 2019, 134: 443-446.

[10] Guo Jing-Jing; Yang Bi-Juan; Jing Chen-Xu; Chen Duo-Zhi; Hao Xiao-Jiang; Rapid synthesis of ismine, a bioactive Amaryllidaceae alkaloid, J Chem Res. 2017, (4): 202-204.

[11] Yuan Wen-Juan; Ding Xiao; Wang Zhe; Yang Bi-Juan; Li Xiao-Nian; Zhang Yu; Chen Duo-Zhi; Li Shun-Lin; Chen Quan; Di Ying-Tong; Aisa Haji Akber; Hao Xiao-Jiang; Two novel diterpenoid heterodimers, Bisebracteolasins A and B, from Euphorbia ebracteolata Hayata, and the cancer chemotherapeutic potential of Bisebracteolasin A, Sci Rep-Uk. 2017, 7.